Description

Technical Parameters

AC-262 99% Raw Material Powder Core Introduction

Pharmaceutical-grade raw material | Made in China AC-262,356 (Selective androgen receptor modulator)

Chemical name : 4-(4-cyanophenoxy)-2-(4-fluorophenyl)-3-(trifluoromethyl)benzamide

CAS No .: 852426-15-2

Molecular formula : C₂₁H₁₂F₄N₂O₂

Molecular weight : 400.33

EINECS ID : Pending Assignment

Melting point : 201-204℃

Appearance : White to off-white crystalline powder

Purity : ≥99% (HPLC detection)

Solubility : Easily soluble in DMSO, slightly soluble in ethanol

Core Function | Core Effects

AC-262 is a highly selective partially agonist androgen receptor modulator (SARM) . Due to its unique trifluoromethylbenzamide structure and partially agonistic properties , it is widely used in the treatment of muscle atrophy, osteoporosis research, and selective androgen regulation .

✅Partial stimulation mechanism :

Tissue selectivity : Exhibits partial agonistic activity in muscle and bone tissues.

Receptor affinity : High affinity for androgen receptors, EC50 < 10 nM

Safety advantages : Partial agonist properties reduce the risk of side effects.

✅Quality advantages of Chinese manufacturing :

Ultra-high purity : Raw material purity ≥ 99%, single impurities ≤ 0.1%

Crystal form control : Stable β-crystal form ensures formulation reproducibility.

Chiral purity : Optical purity of chiral centers ≥ 99.8%

✅Global supply assurance :

Cold chain logistics : constant temperature transportation at 15-25℃ to ensure stability.

Multiple packaging options : 1kg/bag, 5kg/drum, and more.

Customs clearance support : Complete export documents such as MSDS and COA

Production process and quality assurance

1. Advantages of the synthesis process :

Chiral synthesis : Asymmetric synthesis techniques ensure correct chiral center configuration.

Purification process : Column chromatography combined with recrystallization to obtain high-purity crystals.

Drying technology : Vacuum low-temperature drying, moisture content ≤0.5%

2. Strict quality control standards :

Chemical purity :

Main component content: 99.0%~101.0%

Related substances: Single unknown impurity ≤ 0.1%, total impurities ≤ 0.5%

Residual solvent: Complies with ICH Q3C standards

Physical properties :

Particle size distribution: D50 50-100μm

Bulk density: 0.4-0.6 g/cm³

Solubility: Meets the standards for active pharmaceutical ingredients.

3. Stability data :

Long-term stability : Stable for 36 months at 25℃/60%RH.

Accelerated testing : Passed after 6 months at 40℃/75%RH.

Transportation stability : Vibration and drop tests passed.

Scientific Research Applications and Clinical Prospects

1. Research and application areas :

Treatment for muscle atrophy : age-related sarcopenia, cachexia

Osteoporosis : Increases bone density and improves bone quality

Selective androgen regulation : Tissue-selective androgen action

2. Preclinical data :

Moderate efficacy : Animal studies show an 8-12% increase in lean body mass.

Skeletal Improvement : Significantly increased bone mineral density and improved bone biomechanical properties

High safety : partially agonistic properties, low risk of side effects.

3. Key Features and Advantages :

Effective orally : High oral bioavailability, suitable for long-term administration.

Wide therapeutic window : Wide safe dosage range, low risk of side effects

Metabolic stability : Good metabolic stability in the body, with a moderate half-life.

Global supply and service assurance

1. Production capacity :

Annual production capacity : Over 100 kg per year

Flexible manufacturing : Customized specifications and packaging requirements are acceptable.

Production capacity assurance : Multiple production lines ensure stable supply

2. Quality Certification :

System Certification : Certified by ISO 9001 Quality Management System

Compliance with standards : Meets pharmaceutical raw material standards

Complete documentation : Provides a complete package of quality documentation.

3. Logistics support :

Professional Packaging : Triple protection with aluminum foil bag + desiccant + vacuum packaging

Real-time monitoring : Equipped with a temperature and humidity recorder, allowing for full traceability.

Emergency Plan : Establish an emergency response mechanism for abnormal situations.

Why choose the Chinese-made AC-262?

Partial agonist : Partial agonist properties offer greater safety.

Exceptional purity : Over 99% high purity, with strict impurity control.

Advanced technology : Chiral synthesis technique, optical purity up to 99.8%

Reliable supply : Large-scale production capacity, timely delivery

Summarize

AC-262, made in China, is a 99% pure raw material powder representing a high-quality standard for highly safe selective androgen receptor modulators . Through advanced chiral synthesis technology, rigorous quality control, and a stable supply system , it provides high-quality, highly active research raw materials for global research on muscle atrophy and osteoporosis . Choosing Made in China means choosing professional quality and reliable assurance .

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