Description

Technical Parameters

Cagrilintide 5mg/bottle: Key Information

Pharmaceutical -grade peptide formulation | Made in China, Masto peptide (long-acting amylin analogue )

Chemical Name : N-α-Methyl-L-seryl-L-glutamine-L-histyl-L-glutamine-L-arginyl-L-glycyl-L-tyrosyl-L-alanyl-L-alanyl-L-arginyl-L-glutamine-L-phenylalanyl-L-isoleucyl-L-glutamine-L-tryptophanyl-L-leucyl-L-isoleucyl-L-arginyl-L-lysyl-L-glycyl-L-arginyl-glycamide

CAS Number : Pending Assignment (New Molecular Entity)

Specification : 5mg/bottle

Dosage form : Lyophilized powder for injection

Molecular weight : Approximately 4.2 kDa

Appearance : White freeze-dried lumpy powder

Purity : ≥98% (HPLC detection)

Storage conditions : Store at 2-8℃, away from light.

Core Effects

Mastolide is a long-acting amylin analogue that is widely used for the treatment of obesity, management of type 2 diabetes, and improvement of metabolic syndrome due to its unique dual mechanism of action and remarkable weight loss effect .

✅ Dual mechanism of action :

Amylin receptor agonism : Activation of amylin receptors enhances satiety and reduces food intake.

GLP -1 receptor synergy : Synergistically interacts with GLP-1 receptors to enhance weight loss effects.

Long-lasting properties : Fatty acid side chain modification extends the half-life to 7-10 days.

✅ The quality advantages of "Made in China" :

Purity Guaranteed : Solid-phase synthesis process, purity ≥98%, single impurities ≤0.1%

Activity confirmation : In vitro activity EC50 < 0.1 nM, high in vivo potency.

Excellent stability : Accelerated testing showed that the purity remained above 97% for 6 months.

✅ Global supply assurance :

Cold chain logistics : 2-8℃ cold chain transportation throughout the entire process to ensure product stability.

Multi- warehouse delivery : Regional warehouses are established in China, Europe, America, and the Asia-Pacific region, ensuring delivery within 7 days.

Customs clearance support : Professional document preparation ensures smooth customs clearance worldwide.

Production process and quality assurance

1. Advanced synthesis process :

Solid -phase synthesis : Microwave-assisted solid-phase synthesis technology was used, with a condensation efficiency >99.8%.

Fatty acid modification : C18 fatty acid side chain specific modification

Purification process : Preparative HPLC purification, gradient elution, collection of the main peak.

2. Strict quality control standards :

Chemical purity :

Main component content: 98.0%~102.0%

Related substances: Single unknown impurity ≤ 0.1%, total impurities ≤ 0.5%

Acetic acid content: ≤12.0% (ion chromatography)

Biological activity :

Receptor binding assay: Potency not less than 90% of the standard.

In vivo efficacy: Meets quality standards

3. Stability data :

Long-term stability : Stored at 2-8℃ for 24 months, all indicators meet the requirements.

Accelerated testing : After 6 months at 25°C, purity decreased by ≤2.0%.

Stability in use : After reconstitution, store at 2-8℃ for 7 days; purity ≥95%.

Clinical advantages and application prospects

1. Clinical trial data :

Weight loss effect : Phase III clinical trials showed a weight loss of 10-15%.

Blood sugar control : HbA1c decreased by 1.5-2.0%.

Good safety profile : The incidence of adverse events was comparable to that of the control group.

2. Advantages of its mechanism of action :

Dual target : Acts simultaneously on both the amyloid receptor and the GLP-1 receptor.

Synergistic Effect : Dual Mechanisms Produce Synergistic Weight Loss Results

Long-lasting and convenient : Once-weekly dosing improves patient compliance.

3. Application Prospects :

Obesity treatment : Obese patients with a BMI ≥ 30 kg/m² or ≥ 27 kg/m² with complications.

Diabetes Management : Dual Management of Weight and Blood Glucose in Patients with Type 2 Diabetes

Metabolic Improvement : Improves cardiovascular risk factors such as blood lipids and blood pressure.

Global supply and service assurance

1. Supply chain advantages :

Raw material supply : Self-built peptide raw material production base with ample production capacity.

Production Compliance : Passed on-site inspections by NMPA and FDA, and meets international GMP standards.

Quality System : Establish a full traceability system from raw materials to finished products.

2. Logistics Support :

Temperature-controlled packaging : Utilizes phase change materials, maintaining a temperature of 2-8℃ for ≥72 hours.

Real-time monitoring : Equipped with a temperature recorder, temperature data can be traced throughout the entire process.

Emergency Plan : Establish an emergency response mechanism for abnormal situations.

3. Technical Services :

Professional support : Providing technical information and regulatory application support.

Customization service : We can provide customized packaging specifications according to customer needs.

After-sales guarantee : Establish a rapid response mechanism for customer complaints.

Why choose Chinese-made Masdo peptides?

Innovative Mechanism : The first long-acting amylin analog with a dual mechanism of action

Remarkable therapeutic effects : Clinically proven to have significant weight loss and blood sugar lowering effects.

Reliable Quality : Manufactured in strict accordance with international GMP standards, ensuring controllable quality.

Stable supply : A complete supply chain ensures timely and reliable delivery.

Summarize

Made in China, Mastodextrin 5mg lyophilized powder for injection represents a new breakthrough in the treatment of metabolic diseases . Through innovative molecular design, rigorous quality control, and a comprehensive supply chain system , it provides more effective and convenient treatment options for obese and diabetic patients worldwide . Choosing Made in China means choosing innovative quality and reliable assurance .

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