Description

Technical Parameters

STROMUSC brand GW501516 10mg 100 tablets core introduction *

Pharmaceutical grade formulation | STROMUSC brand GW501516 oral tablets

Chemical name : 2-(2-methyl-4-((4-methyl-2-(4-trifluoromethylphenyl)-1,3-thiazo-5-yl)methylthio)phenoxy)acetic acid

CAS No .: 317318-70-0

Specifications : 10mg/tablet, 100 tablets/bottle

Dosage form : Film-coated tablets

Molecular formula : C₂₁H₁₈F₃NO₃S₂

Molecular weight : 453.50

Appearance : White, round, film-coated sheet, engraved with the STROMUSC logo and dividing lines.

Purity : ≥99% (HPLC detection)

Storage conditions : Store at 15-25℃ away from light.

Core Effects

STROMUSC's GW501516 is a highly selective PPARδ agonist that is widely used in metabolic disease research, endurance enhancement, and body composition improvement due to its unique phenoxyacetic acid structure and metabolic regulatory properties .

✅Metabolic regulation mechanism :

PPARδ activation : Selectively activates the PPARδ nuclear receptor, EC50 = 1 nM

Fatty acid oxidation : Enhances fatty acid β-oxidation and promotes lipid metabolism.

Glucose metabolism : Improves insulin sensitivity and regulates glucose metabolism

✅ STROMUSC's unique brand advantages :

Precise dosage : 10mg standard dose, content uniformity RSD ≤ 1.5%

Crystal form control : Stable α-crystal form ensures consistent dissolution.

China cGMP Production : Production strictly adheres to China's cGMP standards.

✅Quality assurance advantages :

Purity Guarantee : Raw material purity ≥ 99.5%, conforming to USP standards.

Dissolution optimization : Dissolution rate ≥ 85% within 30 minutes.

Anti-counterfeiting technologies : holographic anti-counterfeiting labels, QR code traceability system

STROMUSC Brand Quality Advantages

1. Raw material quality control :

Chemical purity : Raw material purity ≥ 99.5% (HPLC detection)

Crystal form control : Stable α-crystal form with consistent solubility.

Impurity control : Single unknown impurity <0.05%, total impurities <0.1%

2. Advantages in formulation technology :

Micronization technology : Raw material particle size D90≤10μm, ensuring rapid dissolution.

Coating system :

Isolation layer: Moisture-proof and oxidation-proof protection

Film coating: Gastric-soluble film coating

Precise dosage : Weight variation of 10mg tablets ≤ ±3%

3. Production Quality System :

cGMP Certification : China's cGMP Certified Production Facilities

Environmental control : Class 100,000 cleanroom, online particle monitoring

Quality Traceability : A Full-Process Electronic Traceability System from Raw Materials to Finished Products

4. Quality control indicators :

Content uniformity : RSD ≤ 1.5% (Pharmacopoeia requirement ≤ 6%)

Dissolution rate : ≥85% dissolution at 30 minutes, ≥90% dissolution at 45 minutes.

Related substances : Degradation products <0.1%, total impurities <0.2%

Stability : Passed accelerated testing after 6 months; shelf life: 36 months.

Application features and advantages

1. Efficacy characteristics :

Endurance Enhancement : Significantly improves aerobic endurance and athletic performance.

Fat reduction : Promotes fat oxidation and improves body composition

Metabolic improvement : Improves blood glucose and lipid metabolism indicators

2. Key Features and Advantages :

High selectivity : 1000 times higher selectivity for PPARδ than for PPARα and PPARγ.

Effective orally : High oral bioavailability and convenient to use.

Good safety profile : Preclinical studies have shown good safety profile.

3. Advantages of use :

Convenient medication use : oral administration, resulting in high patient compliance.

Dosage is flexible : the daily dose of 5-20 mg can be adjusted individually.

Significant effects : Endurance and body composition show marked improvement.

Why choose the STROMUSC brand GW501516 ?

High selectivity : PPARδ selectivity is 1000 times higher than PPARα/γ selectivity.

High purity : Over 99% purity, with strict quality control.

Made in China : Manufactured to cGMP standards, reliable quality

Advanced technology : Micronization technology ensures rapid dissolution

Summary

STROMUSC's GW501516 10mg tablets represent the high-quality standard of highly selective PPARδ agonists . Through advanced manufacturing processes, rigorous quality control, and a stable supply system , STROMUSC provides high-quality, highly active research tools for metabolic disease and sports medicine research worldwide . Choosing STROMUSC means choosing research-grade quality and reliable assurance .

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